MK-0941 free base 是具有⼝服活性的葡糖激酶 (glucokinase) 抑制剂,在葡萄糖浓度为 2.5 和 10 mM 的条件下,对重组⼈ glucokinase 的 EC50 值分别为 240 和 65 nM。MK-0941 free base 具有较强的降⾎糖活性,是 大河
茶馆精加力MK-0941 free base (3 or 10 mg/kg, sing oral dose) treatment reduced blood glucose significantly in db/db Male db/db and db/+ (lean) mice (9-10 weeks of age, weighing 43-45 g) [1].丽音技术www.MedChemExpress diabetes. Diabetes Care. 2011 Dec;34(12):2560-6.
Caution: Product has not been fully validated for medical applications.
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